CRTh2 antagonist 1
CRTh2 antagonist 1 is a CRTh2 antagonist with an IC50 of 89 nM.
Product Specifications
CAS Number
1379445-54-1
UNSPSC
12352005
Hazard Statement
H302-H315-H319-H335
Target
Prostaglandin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Inflammation/Immunology; Endocrinology
Assay Protocol
https://www.medchemexpress.com/2-_5-Methyl-1-_2-_morpholinosulfonyl_benzyl_-3-phenyl-1H-pyrazol-4-yl_acetic_acid.html
Solubility
10 mM in DMSO
Smiles
O=C(O)CC1=C(C)N(CC2=CC=CC=C2S(=O)(N3CCOCC3)=O)N=C1C4=CC=CC=C4
Molecular Formula
C23H25N3O5S
Molecular Weight
455.53
Precautions
P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P403+P233-P405-P501
References & Citations
[1]Andrés M, et al. 2- (1H-Pyrazol-4-yl) acetic acids as CRTh2 antagonists. Bioorg Med Chem Lett. 2013 Jun 1;23 (11) :3349-53.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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