ETA antagonist 1
ETA antagonist 1 is a ETA selective antagonist with an IC50 of 0.08 μM.
Product Specifications
CAS Number
[161801-60-1]
UNSPSC
12352005
Target
Endothelin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/N-_3,4-dimethylisoxazol-5-yl_-5-_pentylamino_naphthalene-1-sulfonamide.html
Solubility
10 mM in DMSO
Smiles
O=S(C1=C2C=CC=C(NCCCCC)C2=CC=C1)(NC3=C(C)C(C)=NO3)=O
Molecular Formula
C20H25N3O3S
Molecular Weight
387.50
References & Citations
[1]Singh S, et al. Structure-Based Inhibitors of Influenza Virus Sialidase. A Benzoic Acid Lead with Novel Interaction. J Med Chem. 1995 Apr 14;38 (8) :1344-54.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
ETA
Curated Selection
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