RXFP3/4 agonist 1
Product Specifications
UNSPSC Description
RXFP3/4 agonist 1 is an agonist of relaxin family peptide 3/4 receptor (RXFP3/4), with EC50s of 82/2 nM, respectivley. RXFP3/4 agonist 1 increases food intake in rats[1].
Target Antigen
RXFP Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/RXFP3-4_agonist_1.html
Solubility
10 mM in DMSO
Smiles
CCC1=C(NC=C2/C=N/NC(NCCC3=CC=C(Cl)C=C3)=N)C2=CC(O)=C1
Molecular Weight
383.87
References & Citations
[1]DeChristopher B, et al. Discovery of a small molecule RXFP3/4 agonist that increases food intake in rats upon acute central administration. Bioorg Med Chem Lett. 2019 Apr 15;29(8):991-994.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-111583/RXFP3-4-agonist-1-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-111583/
Clinical Information
No Development Reported
CAS Number
2351104-40-8
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