GSK894281
GSK894281 is an orally active and highly potent ghrelin receptor full agonist with a pEC50 of [1].
Product Specifications
CAS Number
874958-63-1
UNSPSC
12352005
Target
GHSR
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/gsk894281.html
Solubility
10 mM in DMSO
Smiles
O=S(NC1=CC(N2C[C@H](N[C@H](C2)C)C)=CC=C1OC)(C3=CC(F)=C(C4=CC=C(O4)C)C=C3)=O
Molecular Formula
C24H28FN3O4S
Molecular Weight
473.56
References & Citations
[1]A D Shafton, et al.Oral administration of a centrally acting ghrelin receptor agonist to conscious rats triggers defecation. Neurogastroenterol Motil. 2009 Jan;21 (1) :71-7.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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