ISOX-DUAL
Product Specifications
CAS Number
1962928-22-8
UNSPSC Description
ISOX-DUAL is a dual CBP/BRD4 inhibitor with IC50 values of 0.65 μM and 1.5 μM for CBP and BRD4, respectively[1].
Target Antigen
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/isox-dual.html
Solubility
10 mM in DMSO
Smiles
CC1=C(C2=CC3=C(C=C2)N(CCN4CCOCC4)C(CCC5=CC=C(C=C5)OCCCN(C)C)=N3)C(C)=NO1
Molecular Weight
531.69
References & Citations
[1]Edmonds AK, et, al. Scale-up and optimization of the synthesis of dual CBP/BRD4 inhibitor ISOX-DUAL. Org Biomol Chem. 2022 May 18;20(19):4021-4029.
Shipping Conditions
Room temperature
Clinical Information
No Development Reported
Frequently Asked Questions
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