PK44 (phosphate)
PK44 phosphate is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 value of 15.8 nM[1].
Product Specifications
CAS Number
1017682-66-4
UNSPSC
12352005
Target
Dipeptidyl Peptidase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/pk44-phosphate.html
Solubility
10 mM in DMSO
Smiles
O=P(O)(O)O.FC(F)(C1=NN=C2N1CCN(C(C[C@H](N)CC(C3=CC=C4F)=NNC3=C4F)=O)C2)F
Molecular Formula
C17H19F5N7O5P
Molecular Weight
527.34
References & Citations
[1]Adrian Maddaford, et al. Indazoles for use as dpp-iv inhibitors. WO2008040995A1 (compound 67)
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
DPP-4
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