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CCG-2046

Product Specifications

UNSPSC Description

CCG-2046 is a RGS4 inhibitor with an IC50 of 4.3 μM against RGS4-Gαo interaction signal[1].

Target Antigen

RGS Protein

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

COVID-19-immunoregulation

Field of Research

Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/ccg-2046.html

Solubility

10 mM in DMSO

Smiles

N#CC1(C(C#N)(C#N)C1(C)CCC)C#N

Molecular Weight

198.22

References & Citations

[1]Roman DL, et al. Identification of small-molecule inhibitors of RGS4 using a high-throughput flow cytometry protein interaction assay. Mol Pharmacol. 2007 Jan;71(1):169-75.

Shipping Conditions

Room temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-110054/CCG-2046-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-110054/

Clinical Information

No Development Reported

CAS Number

13017-69-1

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