CCG-2046
CCG-2046 is a RGS4 inhibitor with an IC50 of 4.3 μM against RGS4-Gαo interaction signal[1].
Product Specifications
CAS Number
[13017-69-1]
UNSPSC
12352211
Hazard Statement
H301-H311-H315-H319-H331-H335
Target
RGS Protein
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/ccg-2046.html
Solubility
10 mM in DMSO
Smiles
N#CC1(C(C#N)(C#N)C1(C)CCC)C#N
Molecular Formula
C11H10N4
Molecular Weight
198.22
Precautions
P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P361+P364-P362+P364-P403+P233-P405-P501
References & Citations
[1]Roman DL, et al. Identification of small-molecule inhibitors of RGS4 using a high-throughput flow cytometry protein interaction assay. Mol Pharmacol. 2007 Jan;71 (1) :169-75.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
RGS4
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