Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

GT-2016

GT-2016 is a potent, selective, and brain penetrant histamine H3 receptor antagonist with a Ki of 43.8 nM. GT-2016 displays selectivity against H1 and H2 receptors, and has non-active against histamine methyltransferase[1].

Product Specifications

CAS Number

[152241-24-2]

UNSPSC

12352005

Target

Histamine Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/gt-2016.html

Solubility

10 mM in DMSO

Smiles

O=C(N1CCC(C2=CNC=N2)CC1)CCCCC3CCCCC3

Molecular Formula

C19H31N3O

Molecular Weight

317.47

References & Citations

[1]C E Tedford, et al. Pharmacological characterization of GT-2016, a non-thiourea-containing histamine H3 receptor antagonist: in vitro and in vivo studies. J Pharmacol Exp Ther. 1995 Nov;275 (2) :598-604.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

H3 Receptor

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

Dgcr6 Mouse Gene Knockout Kit (CRISPR)
KN504525 1 Kit

Dgcr6 Mouse Gene Knockout Kit (CRISPR)

Ask
View Details
Uso1 Mouse shRNA Lentiviral Particle (Locus ID 56041)
TL511919V 500 µL Each

Uso1 Mouse shRNA Lentiviral Particle (Locus ID 56041)

Ask
View Details
HINT2 (NM_032593) Human Tagged Lenti ORF Clone
RC208371L3 10 µg

HINT2 (NM_032593) Human Tagged Lenti ORF Clone

Ask
View Details
Anti-Phospho-Serine Polyclonal Antibody
MF-0086960-01 50 µL

Anti-Phospho-Serine Polyclonal Antibody

Ask
View Details
Anti-Phospho-Serine Polyclonal Antibody
MF-0086960-02 100 µL

Anti-Phospho-Serine Polyclonal Antibody

Ask
View Details
Anti-Phospho-Serine Polyclonal Antibody
MF-0086960-03 200 µL

Anti-Phospho-Serine Polyclonal Antibody

Ask
View Details