Tazomeline
Tazomeline is a selective M1 muscarinic receptor agonist. Tazomeline inhibits twitch height in rabbit vas deferens (IC50= 0.001 nM) . Tazomeline can be used for research of neuropsychiatric disorders[1].
Product Specifications
CAS Number
131987-54-7
UNSPSC
12352005
Target
MAChR
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/tazomeline.html
Solubility
10 mM in DMSO
Smiles
CCCCCCSC1=NSN=C1C2=CCCN(C)C2
Molecular Formula
C14H23N3S2
Molecular Weight
297.48
References & Citations
[1]Sauerberg P, et al. Novel functional M1 selective muscarinic agonists. Synthesis and structure-activity relationships of 3- (1,2,5-thiadiazolyl) -1,2,5,6-tetrahydro-1-methylpyridines . J Med Chem. 1992 Jun 12;35 (12) :2274-83.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 1
Available Sizes
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