(S) -ABT-102
(S) -ABT-102 is a TRPV1 Antagonist, with an IC50 of 123 nM. (S) -ABT-102 has analgesic activity[1].
Product Specifications
CAS Number
[808756-70-9]
UNSPSC
12352005
Target
TRP Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Cancer; Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/s-abt-102.html
Purity
99.64
Solubility
10 mM in DMSO
Smiles
O=C(NC1=C2C(NN=C2)=CC=C1)N[C@@H]3C4=CC=C(C(C)(C)C)C=C4CC3
Molecular Formula
C21H24N4O
Molecular Weight
348.44
References & Citations
[1]Gomtsyan A, et al. Identification of (R) -1- (5-tert-butyl-2,3-dihydro-1H-inden-1-yl) -3- (1H-indazol-4-yl) urea (ABT-102) as a potent TRPV1 antagonist for pain management. J Med Chem. 2008 Feb 14;51 (3) :392-5.
Shipping Conditions
Room Temperature
Storage Conditions
Store at room temperature 3 years
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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