Parapenzolate (bromide)

Parapenzolate bromide, an antispasmodic, is an orally active mAChR antagonist. Parapenzolate bromide is an anticholinergic agent[1][2].

Product Specifications

CAS Number

[5634-41-3]

UNSPSC

12352005

Target

MAChR

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/parapenzolate-bromide.html

Solubility

10 mM in DMSO

Smiles

C[N+](CC1)(C)CCC1OC(C(C2=CC=CC=C2)(C3=CC=CC=C3)O)=O.[Br-]

Molecular Formula

C21H26BrNO3

Molecular Weight

420.34

References & Citations

[1]Paris, J., et al. Effect of parapenzolate bromide on the contractility of the gall bladder and sphincter of Oddi. Therapie (1968), 23 (3), 609-18. |[2]Ishimura Yasuko, et al. Pharmacological studies on parapenzolate bromide. 1. Pharmacological studies. Shikoku Igaku Zasshi (1970), 26 (1), 43-51.