PSB-1115 (potassium salt)

PSB-1115 potassium salt is a selective A2B Adenosine Receptor antagonist. PSB-1115 potassium salt inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS) -induced contraction inhibition of acetylcholine (ACh) [1].

Product Specifications

CAS Number

[409344-71-4]

UNSPSC

12352005

Hazard Statement

H302-H315-H319-H335

Target

Adenosine Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

Neuroscience-Neuromodulation

Field of Research

Others

Assay Protocol

https://www.medchemexpress.com/psb-1115-potassium-salt.html

Solubility

10 mM in DMSO

Smiles

O=S(C1=CC=C(C2=NC3=C(NC(N(CCC)C3=O)=O)N2)C=C1)(O[K])=O

Molecular Formula

C14H13KN4O5S

Molecular Weight

388.44

Precautions

P261-P264-P270-P271-P280-P302+P352-P304+P340-P330-P362+P364-P405-P501

References & Citations

[1]Michael S, et al. Adenosine A (2A) agonist and A (2B) antagonist mediate an inhibition of inflammation-induced contractile disturbance of a rat gastrointestinal preparation. Purinergic Signal. 2010 Mar;6 (1) :117-24.