CP-96021 (hydrochloride)
CP-96021 hydrochloride is a balanced, combined, potent and orally active leukotriene D4 (LTD4) /platelet activating factor (PAF) receptor antagonist with Ki values of 34 nM and 37 nM, respectively[1].
Product Specifications
CAS Number
167011-22-5
UNSPSC
12352005
Target
Leukotriene Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/cp-96021-hydrochloride.html
Solubility
10 mM in DMSO
Smiles
CC(N1C2=CC=C(OCC3=CC=CC(/C=C/C4=NC5=CC(F)=CC=C5S4)=C3)C=C2)=NC6=C1C=CN=C6.[H]Cl
Molecular Formula
C29H22ClFN4OS
Molecular Weight
529.03
References & Citations
[1]A. Marfat, et al. The discovery of CP-96,021 and CP-96,486, balanced, combined, potent and orally active leukotriene D4 (LTD4) /platelet activating factor (PAF) receptor antagonists. Bioorganic & Medicinal Chemistry Letters. 1995, 5 (13) : 1377-1382.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
LTC4/CysLT2
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