CGP 54626 (hydrochloride)
CGP 54626 (hydrochloride) is a selective antagonist of GABAB receptor with an IC50 value of 4 nM. CGP 54626 (hydrochloride) can be used to investigate the role of GABAB receptors in neurological signaling[1].
Product Specifications
CAS Number
[149184-21-4]
UNSPSC
12352005
Target
GABA Receptor
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cgp-54626-hydrochloride.html
Purity
99.76
Solubility
10 mM in DMSO
Smiles
O=P(C[C@@H](O)CN[C@H](C1=CC=C(Cl)C(Cl)=C1)C)(CC2CCCCC2)O.Cl
Molecular Formula
C18H29Cl3NO3P
Molecular Weight
444.76
References & Citations
[1]Kaupmann K, et al. GABA (B) -receptor subtypes assemble into functional heteromeric complexes. Nature. 1998 Dec 17;396 (6712) :683-7.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C (Powder, protect from light, stored under nitrogen)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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