SGC2085 (hydrochloride)
SGC2085 hydrochloride is a potent and selective inhibitor of coactivator associated arginine methyltransferase 1 (CARM1) with an IC50 of 50 nM. SGC2085 hydrochloride also selectively inhibits PRMT6 with an IC50 value of 5.2 μM, but not other PRMT proteins[1].
Product Specifications
CAS Number
1821908-49-9
UNSPSC
12352005
Hazard Statement
H315-H319-H320
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/sgc2085-hydrochloride.html
Solubility
10 mM in DMSO
Smiles
[H]Cl.CC1=CC(OC2=CC=C(CNC([C@@H](N)C)=O)C=C2C)=CC(C)=C1
Molecular Formula
C19H25ClN2O2
Molecular Weight
348.87
Precautions
P264-P280-P302+P352-P305+P351+P338-P362
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
PRMT6
Frequently Asked Questions
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