PKMYT1-IN-1
Product Specifications
UNSPSC Description
PKMYT1-IN-1 (Compound 1) is an inhibitor for membrane-associated tyrosine and threonine kinase (PKMYT1), with an IC50 of 8.8 nM. PKMYT1-IN-1 inhibits proliferation of tumor cell HCC1569 with IC50 of 42 nM[1].
Target Antigen
Others
Type
Reference compound
Related Pathways
Others
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/pkmyt1-in-1.html
Solubility
10 mM in DMSO
Smiles
CC1=CC=C(C(C)=C1N2C(N)=C3C(NC4=C(C5=NC=NC2=C53)C=CC=C4)=O)O
Molecular Weight
371.39
References & Citations
[1]Zhu D, et al., Membrane-associated tyrosine and threonine kinase inhibitor and use thereof. WO2024061343A1.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-163490/PKMYT1-IN-1-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-163490/
Clinical Information
No Development Reported
CAS Number
3033609-83-2
Available Sizes
Curated Selection
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