17β-HSD5 inhibitor 1
17β-HSD5 inhibitor 1 (Compound 29) is a potent 17β-HSD5 inhibitor, with an IC50 of 2.9 nM in HEK-293 cells overexpressing human 17β-HSD5[1].
Product Specifications
CAS Number
[243638-37-1]
UNSPSC
12352005
Target
17β-HSD
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Smiles
C[C@@]12[C@]3(CC[C@@]1([H])[C@@]4([H])[C@](C5=CC=CC=C5CC4)([H])CC2)OC(C(C)(CC3)C)=O
Molecular Formula
C24H32O2
Molecular Weight
352.51
References & Citations
[1]Marchais-Oberwinkler S, Henn C, et al. 17β-Hydroxysteroid dehydrogenases (17β-HSDs) as therapeutic targets: protein structures, functions, and recent progress in inhibitor development. J Steroid Biochem Mol Biol. 2011 May;125 (1-2) :66-82.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
More Discoveries
Explore Other Products
Browse additional items from our catalog
RDR-aZGP1-Mu-48Tests 48 Tests
Mouse Alpha-2-Glycoprotein 1, Zinc Binding (aZGP1) ELISA Kit
Sign In for Pricing
View Details 
VAng-Yyj6276-50gEcoli 50 µg (E. coli)
Recombinant Schizosaccharomyces Pombe adg1 Protein (aa 23-166)
Sign In for Pricing
View Details K3007605 3x 1.0 µg
Gm10035 sgRNA CRISPR/Cas9 All-in-One Lentivector set (Mouse)
Sign In for Pricing
View Details