GPR30 agonist-1
GPR30 agonist-1 is a G protein-coupled receptor 30 (GPR30) agonist. GPR30 agonist-1 exerts vasorelaxant effects[1].
Product Specifications
CAS Number
[415919-74-3]
UNSPSC
12352005
Target
Estrogen Receptor/ERR
Type
Reference compound
Related Pathways
Vitamin D Related/Nuclear Receptor
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/gpr30-agonist-1.html
Concentration
10mM
Purity
98.62
Solubility
DMSO : 50 mg/mL (ultrasonic; warming; heat to 80°C)
Smiles
COC(C=C1)=C(C=C1Br)[C@@]2([H])[C@](CC=C3)([H])[C@]3([H])C4=CC(F)=CC=C4N2
Molecular Formula
C19H17BrFNO
Molecular Weight
374.25
References & Citations
[1]Brad R S Broughton, et al. Endothelium-dependent relaxation by G protein-coupled receptor 30 agonists in rat carotid arteries. Am J Physiol Heart Circ Physiol. 2010 Mar;298 (3) :H1055-61.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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