GPR55 agonist 4
GPR55 agonist 4 (Compound 28) is a GPR55 agonist (EC50: 131 nM, and 1.41 nM for hGPR55 and rGPR55) . GPR55 agonist 4 induces β-arrestin recruitment to human GPR55[1].
Product Specifications
CAS Number
3006105-55-8
UNSPSC
12352005
Target
GPR55
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gpr55-agonist-4.html
Purity
98.36
Solubility
DMSO : 100 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
O=C1OC2=CC=C(C3=CN=C(N[C@@H](C4=CC=C(F)C=C4)C)N=N3)C=C2N1C
Molecular Formula
C19H16FN5O2
Molecular Weight
365.36
References & Citations
[1]Hewer RC, et al. Discovery and Characterization of Novel CNS-Penetrant GPR55 Agonists. J Med Chem. 2023 Sep 28;66 (18) :12858-12876.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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