CREBBP-IN-9
CREBBP-IN-9 (Compound 9) is an inhibitor for CREBBP with an Kd of 29 μM[1].
Product Specifications
CAS Number
[1219576-50-7]
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/crebbp-in-9.html
Smiles
O=C(NC1=CC=CC(C(C)=O)=C1)C2=C(SC(C)=C2C)N3N=NN=C3
Molecular Formula
C16H15N5O2S
Molecular Weight
341.39
References & Citations
[1]Xu M, et al., Discovery of CREBBP Bromodomain Inhibitors by High-Throughput Docking and Hit Optimization Guided by Molecular Dynamics. J Med Chem. 2016 Feb 25;59 (4) :1340-9.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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