δ opioid receptor antagonist 1
δ opioid receptor antagonist 1 (compound 6-Cy3) is a fluorescent antagonist probe with high selectivity for δ opioid receptor (DOR) (Ki=1.7 nM) . δ opioid receptor antagonist 1 can be used to study the mechanism of pain perception[1].
Product Specifications
UNSPSC
12171500
Target
Fluorescent Dye; Opioid Receptor
Type
Dye Reagents
Related Pathways
GPCR/G Protein; Neuronal Signaling; Others
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/δ-opioid-receptor-antagonist-1.html
Smiles
OC1=C2O[C@@H]3[C@@]4(C2=C(C[C@@H]5[C@@]4(CC6=C3NC7=C6C=CC=C7NC(CNC(CNC(CNC(CNC(CCCCC[N+]8=C(C(C)(C9=C8C=CC(S(=O)([O-])=O)=C9)C)/C=C/C=C%10N(C%11=C(C/%10(C)C)C=C(S(=O)(O)=O)C=C%11)C)=O)=O)=O)=O)=O)O)C=C1)CCN5CC%12CC%12
Molecular Formula
C64H73N9O14S2
Molecular Weight
1256.45
References & Citations
[1]Drakopoulos, et al. "Design, Synthesis, and Characterization of New δ Opioid Receptor-Selective Fluorescent Probes and Applications in Single-Molecule Microscopy of Wild-Type Receptors." Journal of Medicinal Chemistry (2024) .
Shipping Conditions
Room temperature
Scientific Category
Dye Reagents
Clinical Information
No Development Reported
Isoform
δ Opioid Receptor/DOR
Frequently Asked Questions
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