TS-021 (free base)

DPP-IV-IN-1 is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV), a highly specific serine protease, with an IC50 of 4.6 nM.

Product Specifications

CAS Number

[625110-37-4]

Product Name Alternative

DPP-IV-IN-1

UNSPSC

12352005

Target

Dipeptidyl Peptidase

Type

Reference compound

Related Pathways

Metabolic Enzyme/Protease

Applications

Metabolism-sugar/lipid metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/ts-021-free-base.html

Concentration

10mM

Purity

98.84

Solubility

DMSO : 200 mg/mL (ultrasonic; warming; heat to 60°C)

Smiles

N#C[C@H]1N(C(CNC(C)(C)CO)=O)C[C@@H](F)C1

Molecular Formula

C11H18FN3O2

Molecular Weight

243.28

References & Citations

[1]Fukushima H, et al. Synthesis and structure-activity relationships of potent 4-fluoro-2-cyanopyrrolidine dipeptidyl peptidase IV inhibitors. Bioorg Med Chem. 2008 Apr 1;16 (7) :4093-106.

Shipping Conditions

Blue Ice

Storage Conditions

-20°C, 3 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

DPP-4

Available Sizes

Curated Selection

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