(Rac) -Zevaquenabant
(Rac) -Zevaquenabant ((Rac) -MRI-1867, compound 6b) is a cannabinoid receptor type 1 (CB1R) /iNOS antagonist, with a Ki of 5.7 nM for CB1R. (Rac) -Zevaquenabant is potential for the research of liver fibrosis[1].
Product Specifications
CAS Number
[1610420-28-4]
Product Name Alternative
(Rac) -MRI-1867
UNSPSC
12352005
Target
Cannabinoid Receptor; NO Synthase
Type
Reference compound
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/rac-zevaquenabant.html
Purity
99.20
Solubility
DMSO : 50 mg/mL (ultrasonic)
Smiles
O=S(/N=C(N1N=C(C2=CC=C(Cl)C=C2)C(C3=CC=CC=C3)C1)/N=C(N)/C)(C4=CC=C(C(F)(F)F)C=C4)=O
Molecular Formula
C25H21ClF3N5O2S
Molecular Weight
547.98
References & Citations
[1]Design, Synthesis, and Biological Evaluation of Novel, Non-Brain-Penetrant, Hybrid Cannabinoid CB 1 R Inverse Agonist/Inducible Nitric Oxide Synthase (iNOS) Inhibitors for the Treatment of Liver Fibrosis.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
INOS
Available Sizes
More Discoveries
Explore Other Products
Browse additional items from our catalog
LV711005 1.0 µg DNA
HMGB2 Lentiviral Vector (Human) (CMV) (pLenti-GIII-CMV-GFP-2A-Puro)
Sign In for Pricing
View Details 
RE2606H-01 48 Tests
Human HOXA10 (Homeobox protein Hox-A10) ELISA Kit
Sign In for Pricing
View Details 
RE2606H-02 96 Tests
Human HOXA10 (Homeobox protein Hox-A10) ELISA Kit
Sign In for Pricing
View Details 042465-APC 200 µL
SULT2A1, NT (SULT2A1, HST, STD, Bile salt sulfotransferase, Dehydroepiandrosterone sulfotransferase, Hydroxysteroid Sulfotransferase, ST2, ST2A3, Sulfotransferase 2A1) (APC) discontinued
Sign In for Pricing
View Details