Lusaperidone
Product Specifications
UNSPSC Description
Lusaperidone (R107474) is an α2 adrenergic receptor antagonist with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively.
Target Antigen
Adrenergic Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease; Endocrinology
Assay Protocol
https://www.medchemexpress.com/Lusaperidone.html
Purity
99.81
Solubility
DMSO : 3.45 mg/mL (ultrasonic;warming;heat to 60°C)
Smiles
O=C1C(CCN2CCC(OC3=CC=CC=C34)=C4C2)=C(C)N=C5N1C=CC=C5
Molecular Weight
359.42
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-U00117/Lusaperidone-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-U00117/Lusaperidone-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
214548-46-6
Available Sizes
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