Derazantinib (Racemate)
Derazantinib Racemate (ARQ-087 Racemate) is the racemate of Derazantinib. Derazantinib is an orally bioavailable, ATP competitive tyrosine kinase inhibitor; exhibits potent activity against FGFR1-3 chondrocytes with IC50s of 4.5, 1.8, and 4.5 nM, respectively.
Product Specifications
CAS Number
[2309668-44-6]
Product Name Alternative
ARQ-087 (Racemate)
UNSPSC
12352005
Target
FGFR
Type
Reference compound
Related Pathways
Protein Tyrosine Kinase/RTK
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/Derazantinib_Racemate.html
Concentration
10mM
Purity
99.38
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
COCCNCCC1=CC(NC2=NC=C3CC(C4=CC=CC=C4F)C5=CC=CC=C5C3=N2)=CC=C1
Molecular Formula
C29H29FN4O
Molecular Weight
468.57
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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