CGI 560

CGI 560 is an inhibitor for Bruton's tyrosine kinase (BTK) with an IC50 of 400 nM.

Product Specifications

CAS Number

845269-74-1

UNSPSC

12352005

Target

Btk

Type

Reference compound

Related Pathways

Protein Tyrosine Kinase/RTK

Field of Research

Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/cgi-560.html

Smiles

O=C(C1=CC=C(C(C)(C)C)C=C1)NC2=CC(C3=CN4C(C(NC5=CC=CC=C5)=N3)=NC=C4)=CC=C2

Molecular Formula

C29H27N5O

Molecular Weight

461.56

References & Citations

[1]Lv J, et al., Development of Bruton's Tyrosine Kinase Inhibitors for Rheumatoid Arthritis. Curr Med Chem. 2018;25 (42) :5847-5859.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

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