Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

M617

M617 is a selective galanin receptor 1 (GAL1) agonist, with Kis of 0.23 and 5.71 nM for GAL1 and GAL2, respectively. M617, acting through its central GAL1, can promote GLUT4 expression and enhance GLUT4 content in the cardiac muscle of type 2 diabetic rats[1][2].

Product Specifications

CAS Number

[860790-38-1]

UNSPSC

12352209

Target

Neuropeptide Y Receptor

Type

Peptides

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Cardiovascular Disease

Assay Protocol

https://www.medchemexpress.com/m617.html

Purity

99.54

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

C([C@@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(NCC(N[C@@H](CC1=CC=C(O)C=C1)C(N[C@H](C(N[C@H](C(NCC(=O)N2[C@H](C(N[C@H](C(=O)N3[C@H](C(=O)N4[C@H](C(NCC(N[C@@H](CC5=CC=CC=C5)C(N[C@H](C(=O)N6[C@H](C(N[C@@H](CC7=CC=CC=C7)C(N[C@@H](CCCNC(=N)N)C(N)=O)=O)=O)CCC6)CO)=O)=O)=O)CCC4)CCC3)CCC(N)=O)=O)CCC2)=O)CC(C)C)=O)CC(C)C)=O)=O)=O)C)=O)CO)=O)CC(N)=O)=O)CC(C)C)=O)[C@@H](C)O)=O)NC(CN)=O)C=8C=9C(NC8)=CC=CC9

Molecular Formula

C112H161N29O28

Molecular Weight

2361.65

References & Citations

[1]Lundström, L., et al. A Galanin Receptor Subtype 1 Specific Agonist. Int J Pept Res Ther 11, 17–27 (2005) .|[2]Fang P, et al. Central injection of GalR1 agonist M617 facilitates GLUT4 expression in cardiac muscle of type 2 diabetic rats. Exp Gerontol. 2015;65:85-89.

Shipping Conditions

Blue Ice

Storage Conditions

-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture and light)

Scientific Category

Peptides

Clinical Information

No Development Reported

Available Sizes

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

MGC27016 Antibody
GWB-8DC169 0.05 mg

MGC27016 Antibody

Ask
View Details
RPL36L Antibody
DF9132-01 100 µL

RPL36L Antibody

Ask
View Details
RPL36L Antibody
DF9132-02 200 µL

RPL36L Antibody

Ask
View Details
CPS1 Rabbit pAb
E45R27944N-100 100 µL

CPS1 Rabbit pAb

Ask
View Details
Recombinant Anti-FSTL1 Antibody, Rabbit Monoclonal
MBS8104336-01 0.1 mL

Recombinant Anti-FSTL1 Antibody, Rabbit Monoclonal

Ask
View Details
Recombinant Anti-FSTL1 Antibody, Rabbit Monoclonal
MBS8104336-02 5x 0.1 mL

Recombinant Anti-FSTL1 Antibody, Rabbit Monoclonal

Ask
View Details