SYM 2081
Product Specifications
UNSPSC Description
SYM 2081 is a high-affinity ligand and potent, selective agonist of kainate receptors, inhibits [3H]-kainate binding with an IC50 of 35 nM, almost 3000- and 200-fold selectivity for kainate receptors over AMPA and NMDA receptors respectively[1].
Target Antigen
iGluR
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel;Neuronal Signaling
Applications
Neuroscience-Neurodegeneration
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/sym-2081.html
Purity
98.0
Solubility
H2O : 50 mg/mL (ultrasonic)
Smiles
N[C@@H](C[C@@H](C)C(O)=O)C(O)=O
Molecular Weight
161.16
References & Citations
[1]Lee JY, et al. Furthering pharmacological and physiological assessment of the glutamatergic receptors at the Drosophila neuromuscular junction. Comp Biochem Physiol C Toxicol Pharmacol. 2009 Nov;150(4):546-57.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-101310/SYM-2081-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-101310/SYM-2081-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
31137-74-3
Available Sizes
Curated Selection
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