R-84760
R-84760 is a selective κ-opioid receptor agonist. R-84760 has antinociceptive effect[1][2].
Product Specifications
CAS Number
157824-23-2
UNSPSC
12352005
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/r-84760.html
Smiles
O=C([C@H]1CCC2=C1C=C(Cl)C(Cl)=C2)N3[C@H](CN4CCCC4)CSCC3.Cl
Molecular Formula
C19H25Cl3N2OS
Molecular Weight
435.84
References & Citations
[1]Fujibayashi K, et al. Pharmacological properties of R-84760, a novel kappa-opioid receptor agonist.[J].European Journal of Pharmacology, 1994, 261 (1-2) :133-140.|[2]Fujibayashi K, et al. Profiles of the antinociceptive effect of R-84760, a selective kappa-opioid receptor agonist, in the formalin test in mice. Jpn J Pharmacol. 1995 May;68 (1) :57-63.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 2
Isoform
κ Opioid Receptor/KOR
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