Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

GNE-235

GNE-235 is a compound selective for the second bromodomain of PBRM1, with a KD of 0.28 ± 0.02 μM. GNE-235 can be used for evaluation of the cellular function of PBRM1[1].

Product Specifications

UNSPSC

12352005

Target

Epigenetic Reader Domain

Type

Reference compound

Related Pathways

Epigenetics

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/gne-235.html

Purity

98.45

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

C[C@H]1CCCN1C2=C(N)N=NC(C3=CC=CO3)=C2

Molecular Formula

C13H16N4O

Molecular Weight

244.29

References & Citations

[1]Cochran AG, et al. GNE-235: A Lead Compound Selective for the Second Bromodomain of PBRM1. J Med Chem. 2023 Sep 28;66 (18) :13116-13134.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

Acetyl-Histone H2A (Lys9) Antibody
A10892-100UG 100 µg

Acetyl-Histone H2A (Lys9) Antibody

Ask
View Details
ORF7a protein
PC0001M5 50 µL

ORF7a protein

Ask
View Details
Mouse Siglecl1 Pre-designed siRNA Set B
SI112925B 1 Each

Mouse Siglecl1 Pre-designed siRNA Set B

Ask
View Details
Recombinant Human GMP-PDE gamma/PDE6G (N-His-SUMO)
32-10111-50 50 µg

Recombinant Human GMP-PDE gamma/PDE6G (N-His-SUMO)

Ask
View Details
TAK1L, CT (TAK1L, C21orf7, TAK1-like protein) (MaxLight 490)
MBS6353507-01 0.1 mL

TAK1L, CT (TAK1L, C21orf7, TAK1-like protein) (MaxLight 490)

Ask
View Details
TAK1L, CT (TAK1L, C21orf7, TAK1-like protein) (MaxLight 490)
MBS6353507-02 5x 0.1 mL

TAK1L, CT (TAK1L, C21orf7, TAK1-like protein) (MaxLight 490)

Ask
View Details