LUF5831
LUF5831 is a non-adenosine agonist with an affinity of Ki=18 nM for adenosine A1 receptor[1].
Product Specifications
CAS Number
333963-57-8
UNSPSC
12352005
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/luf5831.html
Smiles
N#CC1=C(SCCO)N=C(C(C#N)=C1C2=CC=C(O)C=C2)N
Molecular Formula
C15H12N4O2S
Molecular Weight
312.35
References & Citations
[1]Heitman LH, et al., Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A1 receptors of LUF5831, a novel nonadenosine-like agonist. Br J Pharmacol. 2006 Mar;147 (5) :533-41.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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