EP300/CBP ligand 1
EP300/CBP ligand 1 is a PROTAC target protein ligand (Ligands for Target Protein for PROTACs) . EP300/CBP ligand 1 can be used for synthesis dCE-2 (HY-161958) [1].
Product Specifications
UNSPSC
12352005
Target
Ligands for Target Protein for PROTAC
Type
Reference compound
Related Pathways
PROTAC
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ep300-cbp-ligand-1.html
Smiles
CN(C=C1)N=C1C2=CC(C(NC3=CC=CC4=C3C=C(C)N=N4)=O)=CC(NC(C)=O)=C2
Molecular Formula
C22H20N6O2
Molecular Weight
400.43
References & Citations
[1]Cheng-Sánchez I, et al. Structure-Based Design of CBP/EP300 Degraders: When Cooperativity Overcomes Affinity. JACS Au. 2024 Aug 8;4 (9) :3466-3474.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
More Discoveries
Explore Other Products
Browse additional items from our catalog
LV754282 1.0 µg DNA
TRNAV4 Lentiviral Vector (Human) (EF1a) (pLenti-GIII-EF1a)
Sign In for Pricing
View Details 
MBS7187618 Inquire
Rabbit anti-Schizosaccharomyces pombe (strain 972/24843)(Fission yeast) RNP24 Polyclonal Antibody
Sign In for Pricing
View Details 
MBS1381447-01 0.02 mg (E-Coli)
Recombinant Clostridium tetani V-type ATP synthase subunit E 1 (atpE1)
Sign In for Pricing
View Details MBS1381447-02 0.1 mg (E-Coli)
Recombinant Clostridium tetani V-type ATP synthase subunit E 1 (atpE1)
Sign In for Pricing
View Details 
MBS1381447-03 0.02 mg (Yeast)
Recombinant Clostridium tetani V-type ATP synthase subunit E 1 (atpE1)
Sign In for Pricing
View Details