K- (D-1-Nal) -FwLL-NH2 (TFA)
K- (D-1-Nal) -FwLL-NH2 TFA is a high affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively) . K- (D-1-Nal) -FwLL-NH2 blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.
Product Specifications
UNSPSC
12352209
Target
GHSR
Type
Peptides
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/k-d-1-nal-fwll-nh2-tfa.html
Solubility
10 mM in DMSO
Smiles
CC(C)C[C@@H](C(N)=O)NC([C@H](CC(C)C)NC([C@@H](CC1=CNC2=C1C=CC=C2)NC([C@H](CC3=CC=CC=C3)NC([C@@H](CC4=C5C=CC=CC5=CC=C4)NC([C@H](CCCCN)N)=O)=O)=O)=O)=O.O=C(O)C(F)(F)F
Molecular Formula
C53H68F3N9O8
Molecular Weight
1016.16
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Frequently Asked Questions
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