CP59430
CP59430 is an azide analog of the α-adrenaline receptor antagonist Prazosin. P59430 behaves as a competitive antagonist of α1-adrenaline receptor before photolysis. After photolysis, it specifically and irreversibly labels α1-adrenaline receptor and exhibits non-competitive antagonist activity. CP59430 can be used for the study of receptor molecular characterization[1].
Product Specifications
CAS Number
86329-06-8
UNSPSC
12352005
Target
Adrenergic Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Endocrinology
Assay Protocol
https://www.medchemexpress.com/cp59430.html
Smiles
COC1=CC2=NC(N3CCN(C(C4=CC=C(N=[N+]=[N-])C=C4)=O)CC3)=NC(N)=C2C=C1OC
Molecular Formula
C21H22N8O3
Molecular Weight
434.45
References & Citations
[1]Hess, et al. "Photoaffinity label for the alpha 1-adrenergic receptor: synthesis and effects on membrane and affinity-purified receptors." Proceedings of the National Academy of Sciences 80.8 (1983) : 2102-2106.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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