Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

JNJ-31020028

JNJ-31020028 is a selective and brain penetrant antagonist of neuropeptide Y Y2 receptor with pIC50 values of 8.07 and 8.22 for human and rat Y2 receptor, respectively. JNJ-31020028 can be used for the research of nervous disease[1].

Product Specifications

CAS Number

1094873-14-9

UNSPSC

12352005

Hazard Statement

H302, H315, H319, H335

Target

Neuropeptide Y Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease; Endocrinology

Assay Protocol

https://www.medchemexpress.com/JNJ-31020028.html

Concentration

10mM

Purity

98.02

Solubility

DMSO : 21.5 mg/mL (ultrasonic; warming)

Smiles

O=C(N(CC)CC)C(N1CCN(C2=CC=C(NC(C3=C(C4=CC=CN=C4)C=CC=C3)=O)C=C2F)CC1)C5=CC=CC=C5

Molecular Formula

C34H36FN5O2

Molecular Weight

565.68

Precautions

H302, H315, H319, H335

References & Citations

[1]Shoblock JR, et al. In vitro and in vivo characterization of JNJ-31020028 (N- (4-{4-[2- (diethylamino) -2-oxo-1-phenylethyl]piperazin-1-yl}-3-fluorophenyl) -2-pyridin-3-ylbenzamide), a selective brain penetrant small molecule antagonist of the neuropeptide Y Y (2) receptor. Psychopharmacology (Berl) . 2010 Feb;208 (2) :265-77.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

NPY Y2 receptor

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

LZTFL1 Human Gene Knockout Kit (CRISPR)
KN207289LP 1 Kit

LZTFL1 Human Gene Knockout Kit (CRISPR)

Sign In for Pricing
View Details
Histone H3 (Ab-9) Antibody
8D0026-AAT 50 µg

Histone H3 (Ab-9) Antibody

Sign In for Pricing
View Details
Human SYDE2 activation kit by CRISPRa
GA113392 1 Kit

Human SYDE2 activation kit by CRISPRa

Sign In for Pricing
View Details
N,N'-Diphenylformamidine
TRC-D491000-50G 50 g

N,N'-Diphenylformamidine

Sign In for Pricing
View Details
C8 (C8G) Rabbit Polyclonal Antibody
TA369568 100 µL

C8 (C8G) Rabbit Polyclonal Antibody

Sign In for Pricing
View Details
QDPR Antibody
KC-46552-01 50 μL

QDPR Antibody

Sign In for Pricing
View Details