Dynorphin A (1-8)
Dynorphin A (1-8) is the predominant opioid peptide identified in placental tissue extracts. Dynorphin A (1-8) is the most likely natural ligand of the kappa receptor. The binding of 3H-Bremazocine to the purified kappa receptor is inhibited by Dynorphin A (1-8) (IC50=303 nM) [1][2].
Product Specifications
CAS Number
75790-53-3
UNSPSC
12352209
Target
Endogenous Metabolite; Opioid Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Metabolic Enzyme/Protease; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/dynorphin-a-1-8.html
Purity
99.88
Solubility
10 mM in DMSO
Smiles
Molecular Formula
C46H72N14O10
Molecular Weight
981.15
References & Citations
Shipping Conditions
Blue Ice
Storage Conditions
-80°C, 2 years; -20°C, 1 year (Powder, stored under nitrogen, away from moisture)
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
Human Endogenous Metabolite; κ Opioid Receptor/KOR
Available Sizes
Frequently Asked Questions
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