Ersentilide
Product Specifications
UNSPSC Description
Ersentilide, a benzamide derivative, is a is a β1-adrenoceptor antagonist and Ikr blocker. Ersentilide is effective in several intact animal models of arrhythmia[1][2].
Target Antigen
Adrenergic Receptor; Potassium Channel
Type
Reference compound
Related Pathways
GPCR/G Protein;Membrane Transporter/Ion Channel;Neuronal Signaling
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/ersentilide.html
Smiles
CS(NC(C=C1)=CC=C1OC[C@@H](O)CNCCOC2=CC=C(N3C=CN=C3)C=C2)(=O)=O
Molecular Weight
446.52
References & Citations
[1]Adamson PB, et, al. Antifibrillatory efficacy of ersentilide, a novel beta-adrenergic and Ikr blocker, in conscious dogs with a healed myocardial infarction. Cardiovasc Res. 1998 Oct;40(1):56-63.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-167866/Ersentilide-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-167866/
Clinical Information
No Development Reported
CAS Number
125279-79-0
Curated Selection
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