Ersentilide
Ersentilide, a benzamide derivative, is a is a β1-adrenoceptor antagonist and Ikr blocker. Ersentilide is effective in several intact animal models of arrhythmia[1][2].
Product Specifications
CAS Number
125279-79-0
UNSPSC
12352005
Target
Adrenergic Receptor; Potassium Channel
Type
Reference compound
Related Pathways
GPCR/G Protein; Membrane Transporter/Ion Channel; Neuronal Signaling
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/ersentilide.html
Smiles
CS(NC(C=C1)=CC=C1OC[C@@H](O)CNCCOC2=CC=C(N3C=CN=C3)C=C2)(=O)=O
Molecular Formula
C21H26N4O5S
Molecular Weight
446.52
References & Citations
[1]Adamson PB, et, al. Antifibrillatory efficacy of ersentilide, a novel beta-adrenergic and Ikr blocker, in conscious dogs with a healed myocardial infarction. Cardiovasc Res. 1998 Oct;40 (1) :56-63.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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