(S) -Gebr32a
(S) -Gebr32a is a potent PDE4 inhibitor with IC50 values of 19.5, 2.1 µM for PDE4 cat; PDE4D3, respectively[1].
Product Specifications
CAS Number
3055162-32-5
UNSPSC
12352005
Target
Phosphodiesterase (PDE)
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/s-gebr32a.html
Smiles
FC(F)OC1=CC=C(C2=NN(C[C@@H](O)CN3CCOCC3)C=C2)C=C1OC4CCCC4
Molecular Formula
C22H29F2N3O4
Molecular Weight
437.48
References & Citations
[1]Cavalloro V, et al. Insight into GEBR-32a: Chiral Resolution, Absolute Configuration and Enantiopreference in PDE4D Inhibition. Molecules. 2020 Feb 19;25 (4) :935.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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