Bilaid C

Bilaid C, a tetrapeptide, can be isolated from the Australian estuarine isolate of Penicillium sp. MST-MF667. Bilaid C is also a potent and selective μ-Opioid Receptor (MOPr) agonist (Ki=210 nM, hMOPr) [1].

Product Specifications

CAS Number

[2393866-13-0]

UNSPSC

12352209

Target

Opioid Receptor

Type

Peptides

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/bilaid-c.html

Solubility

10 mM in DMSO

Smiles

OC(C=C1)=CC=C1C[C@H](N)C(N[C@H](C(C)C)C(N[C@@H](C(C)C)C(N[C@@H](C(O)=O)CC2=CC=CC=C2)=O)=O)=O

Molecular Formula

C28H38N4O6

Molecular Weight

526.62

References & Citations

[1]Dekan Z, et al. A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptor. Proc Natl Acad Sci U S A. 2019 Oct 29;116 (44) :22353-22358.