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PRL3-CNNM4 PPI-IN-1

PRL3-CNNM4 PPI IN 1 (Compound C28d52) is an inhibitor of the PRL3-CNNM4 interaction and also inhibits PRL-mediated suppression of CNNM. PRL3-CNNM4 PPI IN 1 is capable of penetrating epithelial cell layers, exhibits metabolic stability, possesses favorable pharmacokinetic and pharmacodynamic properties, and holds potential for drug development based on this compound[1].

Product Specifications

CAS Number

[40133-06-0]

UNSPSC

12352005

Hazard Statement

H302, H315, H319, H335

Target

Phosphatase

Type

Reference compound

Related Pathways

Metabolic Enzyme/Protease

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/prl3-cnnm4-interaction-in-1.html

Purity

99.33

Smiles

O=C(O)C1=CC2=C(S1)CCC2

Molecular Formula

C8H8O2S

Molecular Weight

168.21

Precautions

H302, H315, H319, H335

References & Citations

[1]Funato Y, et al. Development of a high-throughput screening system targeting the protein-protein interactions between PRL and CNNM[J]. Scientific Reports, 2024, 14 (1) : 25432.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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