Carbinoxamine-d6 (maleate)
Carbinoxamine-d6 (maleate) is the deuterium labeled Carbinoxamine maleate salt. Carbinoxamine maleate salt is a histamine H1 receptor antagonist.
Product Specifications
UNSPSC
12352005
Target
Histamine Receptor; Isotope-Labeled Compounds
Type
Isotope-Labeled Compounds
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling; Others
Field of Research
Neurological Disease; Endocrinology
Solubility
10 mM in DMSO
Smiles
ClC1=CC=C(C(C2=NC=CC=C2)OCCN(C([2H])([2H])[2H])C([2H])([2H])[2H])C=C1.O=C(O)/C=C\C(O)=O
Molecular Formula
C20H17D6ClN2O5
Molecular Weight
412.90
References & Citations
[1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53 (2) :211-216. |[2]Harikrishnan A, et al. The cooperative effect of Lewis pairs in the Friedel-Crafts hydroxyalkylation reaction: a simple and effective route for the synthesis of (±) -carbinoxamine. Org Biomol Chem. 2015 Mar 28;13 (12) :3633-47.
Shipping Conditions
Room temperature
Scientific Category
Isotope-Labeled Compounds
Clinical Information
No Development Reported
Isoform
H1 Receptor
Available Sizes
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