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Terevalefim

Product Specifications

UNSPSC Description

Terevalefim (ANG-3777), an hepatocyte growth factor (HGF) mimetic, selectively activates the c-Met receptor[1][2].

Target Antigen

c-Met/HGFR

Type

Reference compound

Related Pathways

Protein Tyrosine Kinase/RTK

Field of Research

Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/terevalefim.html

Smiles

C1(/C=C/C2=CC=CS2)=NNC=C1

Molecular Weight

176.24

References & Citations

[1]Jonathan S Bromberg, et al. Renal Function Improvement Following ANG-3777 Treatment in Patients at High Risk for Delayed Graft Function After Kidney Transplantation. Transplantation. 2021 Feb 1;105(2):443-450.|[2]Latha Paka, et al. The Effect of ANG-3777 on Hepatocyte Growth Factor Receptor, c-MET Signaling. American Transplant Society.

Shipping Conditions

Room Temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-137455/Terevalefim-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-137455/Terevalefim-SDS-MedChemExpress.pdf

CAS Number

1070881-42-3

Available Sizes

Curated Selection

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