Anticonvulsant agent 5
Anticonvulsant agent 5 (Compound 5c) exhibits high affinity for GABAA receptors and NaV1.3 receptors. Anticonvulsant agent 5 shows anticonvulsant efficacy in mice psychomotor epilepsy test with an ED50 of 107 mg/kg. Anticonvulsant agent 5 exhibits neuroprotective activity against Kainic acid with an IC50 of 113 μM. Anticonvulsant agent 5 is blood-brain barrier (BBB) penetrable[1].
Product Specifications
CAS Number
9007-83-4
UNSPSC
12352005
Target
GABA Receptor; Sodium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/anticonvulsant-agent-5.html
Smiles
S=C1N(C2=CC=C(OC)C=C2)C(C(NC(C3=CC=C(F)C=C3)=O)CC4=CC=CC=C4)=NN1
Molecular Formula
C24H21FN4O2S
Molecular Weight
448.51
References & Citations
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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