Isotodesnitazene
Product Specifications
UNSPSC Description
Isotodesnitazene is a kind of opioids. Isotodesnitazene primarily acts on μ-opioid receptors (MOR). Isotodesnitazene has an EC50 of 34.8 nM for MOR-βarr2 and 142 nM for MOR-mini-Gi. Isotodesnitazene can be used in the study of opioids[1].
Target Antigen
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling
Field of Research
Metabolic Disease; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/isotodesnitazene.html
Solubility
DMSO : ≥ 100 mg/mL
Smiles
CC(C)OC(C=C1)=CC=C1CC2=NC3=C(N2CCN(CC)CC)C=CC=C3
Molecular Weight
365.51
References & Citations
[1]Vandeputte MM, et al. Synthesis, Chemical Characterization, and μ-Opioid Receptor Activity Assessment of the Emerging Group of "Nitazene" 2-Benzylbenzimidazole Synthetic Opioids. ACS Chem Neurosci. 2021 Apr 7;12(7):1241-1251.
Shipping Conditions
Room Temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-164747/Isotodesnitazene-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-164747/Isotodesnitazene-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
2732926-27-9
Available Sizes
Curated Selection
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