Perlapine
Product Specifications
UNSPSC Description
Perlapine is a potent muscarinic DREADD (Designer Receptors Exclusively Activated by Designer agents) agonist Perlapine exhibits >10000-fold selectivity for hM3Dq over hM3 receptors[1].
Target Antigen
mAChR
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/perlapine.html
Solubility
10 mM in DMSO
Smiles
CN1CCN(C2=NC(C=CC=C3)=C3CC4=CC=CC=C24)CC1
Molecular Weight
291.39
References & Citations
[1]Chen X, et al. The first structure-activity relationship studies for designer receptors exclusively activated by designer drugs. ACS Chem Neurosci. 2015 Mar 18;6(3):476-84.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-110239/Perlapine-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-110239/
Clinical Information
No Development Reported
CAS Number
1977-11-3
Available Sizes
Curated Selection
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