Perlapine
Perlapine is a potent muscarinic DREADD (Designer Receptors Exclusively Activated by Designer agents) agonist Perlapine exhibits >10000-fold selectivity for hM3Dq over hM3 receptors[1].
Product Specifications
CAS Number
1977-11-3
Product Name Alternative
MP-11
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H413
Target
MAChR
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/perlapine.html
Purity
99.6
Solubility
10 mM in DMSO
Smiles
CN1CCN(C2=NC(C=CC=C3)=C3CC4=CC=CC=C24)CC1
Molecular Formula
C19H21N3
Molecular Weight
291.39
Precautions
H302, H315, H319, H413
References & Citations
[1]Chen X, et al. The first structure-activity relationship studies for designer receptors exclusively activated by designer drugs. ACS Chem Neurosci. 2015 Mar 18;6 (3) :476-84.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
GTR15311834 1 Vial
Lentiviral human ITSN1 shRNA (UAS) - Lentiviral human ITSN1 shRNA (UAS, RFP) (25)
Sign In for Pricing
View Details LV686130 1.0 µg DNA
MGLL Lentiviral Vector (Rat) (EF1a) (pLenti-GIII-EF1a)
Sign In for Pricing
View Details GTR15107382 1 Vial
Lentiviral human KIN shRNA (UAS) - Lentiviral human KIN shRNA (UAS) (100)
Sign In for Pricing
View Details NBP3-05916F 0.1 mL
Rabbit Monoclonal Serpin B6 Antibody (202) [FITC]
Sign In for Pricing
View Details