PIN1 inhibitor 3
Product Specifications
UNSPSC Description
PIN1 inhibitor 3 (Compound A0) is a PIN1 inhibitor, with a KD of 25 nM and an IC50 of 150 nM. PIN1 inhibitor 3 can be used as a target protein ligand for the synthesis of PROTAC. PIN1 inhibitor 3 can be utilized in cancer research[1].
Target Antigen
Ligands for Target Protein for PROTAC; PIN1
Type
Reference compound
Related Pathways
PI3K/Akt/mTOR;PROTAC
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/pin1-inhibitor-3.html
Smiles
CC1=CC=CC=C1C2(CC2)C(NC(C(NC(CC3)CCN3C)=O)CC(N=N4)=CN4C(C=C5)=CC=C5C(C=C6)=CC=C6C#N)=O
Molecular Weight
587.71
References & Citations
[1]Liu C, et al. Re-Evaluating PIN1 as a Therapeutic Target in Oncology Using Neutral Inhibitors and PROTACs. J Med Chem. 2024 Sep 12;67(17):15780-15795.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-168036/PIN1-inhibitor-3-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-168036/
Clinical Information
No Development Reported
CAS Number
3039570-04-9
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
![Mouse Monoclonal CD45RB Antibody (BRA-11 (same as BRA-11G)) [Janelia Fluor 646]](https://cdn.genprice.uk/genprice/genprice2.png)
NBP2-34564JF646 0.1 mL
Mouse Monoclonal CD45RB Antibody (BRA-11 (same as BRA-11G)) [Janelia Fluor 646]
Ask
View Details