NS-2710
NS-2710 is a high-efficacy GABAAα3 agonist with a Ki of 9.2 nM. NS-2710 can be used for anxiety research[1].
Product Specifications
CAS Number
[184220-36-8]
UNSPSC
12352005
Target
GABA Receptor
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ns-2710.html
Purity
99.21
Solubility
DMSO : 13.16 mg/mL (ultrasonic)
Smiles
C/C(C1=CC=C2C(N=CN2C3=CC=CC(C4=CC=CN=C4)=C3)=C1)=N\OCC
Molecular Formula
C22H20N4O
Molecular Weight
356.42
References & Citations
[1]John R Atack. GABAA receptor subtype-selective modulators. I. α2/α3-selective agonists as non-sedating anxiolytics. Curr Top Med Chem. 2011;11 (9) :1176-202.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 2
Available Sizes
Curated Selection
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