PD-151307
PD-151307 is an N-type calcium channel antagonist with significant inhibitory effects in IMR-32 human neuroblastoma cells, exhibiting an IC50 of 0.32 µM. PD-151307 can be used in research related to cancer therapy, anticonvulsants, and neuropathic pain[1].
Product Specifications
CAS Number
[225925-12-2]
UNSPSC
12352005
Target
Calcium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Field of Research
Cancer; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/pd-151307.html
Smiles
O=C([C@@H](NC([C@@H](NC(N1CCCCCC1)=O)CC(C)C)=O)CC2=CC=C(C=C2)OCC3=CC=CC=C3)OC(C)(C)C
Molecular Formula
C33H47N3O5
Molecular Weight
565.74
References & Citations
[1]Hu LY, et al. N, N-dialkyl-dipeptidylamines as novel N-type calcium channel blockers. Bioorg Med Chem Lett. 1999 Mar 22;9 (6) :907-12.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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